Journal of Medicinal Chemistry
Volume 41, Issue 8 (April 9, 1998)
Copyright © 1998
American Chemical Society
| COMMUNICATIONS TO THE EDITOR | |
1205-1208 | 4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]- piperazinyl]-6,7-dimethoxyquinazoline (L-765,314): A Potent and Selective  1b Adrenergic Receptor Antagonist
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ARTICLES | |
1209-1217 | Inhibition of Membrane-Type 1 Matrix Metalloproteinase by Hydroxamate Inhibitors: An Examination of the Subsite Pocket
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1218-1235 | The Selective 5-HT1B Receptor Inverse Agonist 1'-Methyl-5-[[2'-methyl-4'- (5-methyl-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) Potently Blocks Terminal 5-HT Autoreceptor Function Both in Vitro and in Vivo
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1236-1241 | Synthesis and Antiviral Evaluation of Certain Novel Pyrazinoic Acid C-Nucleosides
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1242-1251 | Design, Synthesis, and Antiviral Activity of -Nucleosides: D- and L-Isomers of Lyxofuranosyl- and (5-Deoxylyxofuranosyl)benzimidazoles
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1252-1262 | Design, Synthesis, and Antiviral Evaluations of 1-(Substituted benzyl)-2-substituted-5,6-dichlorobenzimidazoles as Nonnucleoside Analogues of 2,5,6-Trichloro-1-( -D-ribofuranosyl)benzimidazole
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1263-1271 | Selective Pneumocystis carinii Dihydrofolate Reductase Inhibitors: Design, Synthesis, and Biological Evaluation of New 2,4-Diamino-5-substituted-furo[2,3-d]pyrimidines
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1272-1283 | Synthesis and Pharmacology of Conformationally Restricted Raloxifene Analogues: Highly Potent Selective Estrogen Receptor Modulators
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1284-1298 | Synthesis and Antiviral Activity of Novel Acyclic Nucleosides: Discovery of a Cyclopropyl Nucleoside with Potent Inhibitory Activity against Herpesviruses
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1299-1305 | d-Fused [1]Benzazepines with Selective in Vitro Antitumor Activity: Synthesis and Structure-Activity Relationships
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1306-1314 | Epidoxoform: A Hydrolytically More Stable Anthracycline-Formaldehyde Conjugate Toxic to Resistant Tumor Cells
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1315-1343 | Structure-Activity Studies on Anticonvulsant Sugar Sulfamates Related to Topiramate. Enhanced Potency with Cyclic Sulfate Derivatives
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1344-1351 | Azapeptides as Inhibitors and Active Site Titrants for Cysteine Proteinases
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BOOK REVIEWS | |
1352-1353 | Protein Structure: A Practical Approach Edited by T. E. Creighton, Editor. IRL Press, New York. 1997. xxiii + 383 pp. 15.5 x 23.5 cm. ISBN 0-19-963618-4. $55.00 (pbk). Protein Function: A Practical Approach Edited by T. E. Creighton, Editor. IRL Press, New York. 1997. xxi + 334 pp. 15.5 x 23.5 cm. ISBN 0-19-963615-4. $55.00 (pbk).
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1353-1353 | Guanidino Compounds in Biology and Medicine: 2 Edited by P. De Deyn, B. Mareseau, I. A. Quneshi, and A. Mori. John Libbey & Company Limited, London. 1997. 405 pp. 19.5 × 24.5 cm. ISBN 0-81696-543-4.  66.00.
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1353-1354 | Antiviral Chemotherapy By Richard Challand and Robert J. Young. In Biochemical and Medicinal Chemistry Series. Series Editor John Mann. Spektrum Academic Publishers, Oxford, and University Science Books, Sausolito. 1997. viii + 128 pp. 19 × 24.5 cm. ISBN 1-901217-03-5. $28.50 (pbk).
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1354-1354 | Introduction to Medicinal Chemistry: How Drugs Act and Why Alex Gringauz. Wiley-VCH, Inc., New York. 1997. xiii + 721 pp. 18.5 × 26 cm. ISBN 0-471-18545-0. $89.95.
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1354-1355 | Annual Reports in Combinatorial Chemistry and Molecule Diversity, Volume 1 Edited by Walter H. Moos, Michael R. Pavia, Andrew D. Ellington, and Brian K. Kay. ESCOM Publishers, Leiden, The Netherlands. 1997. xiii + 354 pp. 17 × 24.5 cm. ISBN 90-72199-23.5. $97.00.
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1355-1356 | Purinergic Approaches in Experimental Therapeutics Edited by Kenneth A. Jacobson and Michael F. Jarvis. Wiley-Liss, New York. 1997. xiv + 581 pp. 16 × 24 cm. ISBN 0-47114071-6. $89.95.
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